From the Promiscuous Asenapine to Potent Fluorescent Ligands Acting at a Series of Aminergic G-Protein-Coupled Receptors

Candide Hounsou (1) , Corinne Baehr (2) , Vincent Gasparik (2) , Doria Alili (1) , Abderazak Belhocine (1) , Thieric Rodriguez (1) , Elodie Dupuis (3) , Thomas Roux (3) , André Mann (2) , Denis Heissler (2, 4) , Jean-Philippe Pin (1) , Thierry Durroux (1) , Dominique Bonnet (2, 4) , Marcel Hibert (2, 4)

1 IGF - Institut de Génomique Fonctionnelle
2 LIT - Laboratoire d'Innovation Thérapeutique
3 Cisbio Bioassays
4 Centre de recherche du médicament Medalis - Drug Discovery Center [LabEx]

Domaines: Chimie; Chimie thérapeutique

Candide Hounsou, Corinne Baehr, Vincent Gasparik, Doria Alili, Abderazak Belhocine, et al.. From the Promiscuous Asenapine to Potent Fluorescent Ligands Acting at a Series of Aminergic G-Protein-Coupled Receptors. Journal of Medicinal Chemistry, 2017, 61 (1), pp.174-188. ⟨10.1021/ACS.JMEDCHEM.7B01220⟩. ⟨hal-02366277⟩