Carbonic anhydrase inhibitors : comparison of aliphatic sulfamate/bis-sulfamate adducts with isozymes II and IX as a platform for designing tight-binding, more isoform-selective inhibitors

Rosa Maria Vitale (1) , Vincenzo Alterio (1) , Alessio Innocenti (2) , Jean-Yves Winum (3) , Simona Maria Monti (1) , Giuseppina de Simone (1) , Claudiu T. Supuran (2)

1 Istituto di Biostructure e Bioimmagini
2 LCBI-UniFI - Laboratorio di Chimica Bioinorganica [UniFI, Firenze] = Laboratory of Bioinorganic Chemistry [UniFI Florence]
3 IBMM - Institut des Biomolécules Max Mousseron [Pôle Chimie Balard]

Domaines: Chimie organique

Rosa Maria Vitale, Vincenzo Alterio, Alessio Innocenti, Jean-Yves Winum, Simona Maria Monti, et al.. Carbonic anhydrase inhibitors : comparison of aliphatic sulfamate/bis-sulfamate adducts with isozymes II and IX as a platform for designing tight-binding, more isoform-selective inhibitors. Journal of Medicinal Chemistry, 2009, 52 (19), pp.5990-5998. ⟨10.1021/jm900641r⟩. ⟨hal-00460022⟩