Carbonic anhydrase inhibitors: Binding of an antiglaucoma glycosyl-sulfanilamide derivative to human isoform II and its consequences for the drug design of enzyme inhibitors incorporating sugar moieties

Anna Di Fiore (1) , Claudiu T. Supuran (2) , Jean-Yves Winum (3) , Jean-Louis Montero (3) , Carlo Pedone (1, 4) , Andrea Scozzafava (2) , Giuseppina de Simone (1)

1 Istituto di Biostructure e Bioimmagini
2 LCBI-UniFI - Laboratorio di Chimica Bioinorganica [UniFI, Firenze] = Laboratory of Bioinorganic Chemistry [UniFI Florence]
3 IBMM - Institut des Biomolécules Max Mousseron [Pôle Chimie Balard]
4 Dipartimento delle Scienze Biologiche-Sezione Biostructure

Domaines: Chimie organique

Anna Di Fiore, Claudiu T. Supuran, Jean-Yves Winum, Jean-Louis Montero, Carlo Pedone, et al.. Carbonic anhydrase inhibitors: Binding of an antiglaucoma glycosyl-sulfanilamide derivative to human isoform II and its consequences for the drug design of enzyme inhibitors incorporating sugar moieties. Bioorganic and Medicinal Chemistry Letters, 2007, 17, pp.1726-1731. ⟨10.1016/j.bmcl.2006.12.099⟩. ⟨hal-00273199⟩