The world of [beta]-and [gamma]-peptides comprised of homologated proteinogenic amino acids and other components, Chem. Biodivers, vol.31, pp.1111-1239, 1997. ,
NMR determination of the major solution conformation of a peptoid pentamer with chiral side chains, Proc. Nat. Acad. Sci. U.S.A, vol.95, pp.13525-13530, 1998. ,
Solvophobically Driven Folding of Nonbiological Oligomers, Science, vol.277, pp.1793-1796, 1997. ,
Designed Self-Generation of an Extended Helical Structure From an Achiral Polyheterocylic Strand, Angew. Chem. Int. Ed, vol.118, pp.1845-1847, 1996. ,
Aromatic delta-peptides: design, synthesis and structural studies of helical, quinoline-derived oligoamide foldamers, European Journal of Organic Chemistry, vol.59, pp.17-29, 2003. ,
, Rule of five in 2015 and beyond: Target and ligand structural limitations, ligand chemistry structure and drug discovery project decisions, vol.101, pp.34-41, 2016.
Systematic analysis of helical protein interfaces reveals targets for synthetic inhibitors, ACS Chem. Biol, vol.5, pp.919-923, 2010. ,
Stabilized helical peptides: overview of the technologies and therapeutic promises, Exp. Opin. Drug Discov, vol.6, pp.937-963, 2011. ,
, Peptides: from structure to function, vol.101, pp.3219-3232, 2001.
Application of alicyclic beta-amino acids in peptide chemistry, Chem Soc Rev, vol.35, pp.323-334, 2006. ,
Probing the helical secondary structure of short-chain [beta]-peptides, Helv. Chim. Acta, vol.79, pp.2043-2066, 1996. ,
Synthesis and Characterization of trans-2-Aminocyclohexanecarboxylic Acid Oligomers: An Unnatural Helical Secondary Structure and Implications for beta-Peptide Tertiary Structure, J. Am. Chem. Soc, vol.118, pp.2711-2718, 1996. ,
Evidence that the ?-Peptide 14-Helix is Stabilized by ?3-Residues with Side-Chain Branching Adjacent to the ?-Carbon Atom, Relationship between Side Chain Structure and 14-Helix Stability of ?3-Peptides in Water, vol.85, pp.167-178, 2002. ,
Mixed ?2/?3-Hexapeptides and ?2/?3-Nonapeptides Folding to (P)-Helices with Alternating Twelve-and Ten-Membered Hydrogen-Bonded Rings, Helv. Chim. Acta, vol.80, pp.2577-2593, 1997. ,
Robust mixed 10/12 helices promoted by "alternating chirality" in a new family of C-linked carbo-beta-peptides, J. Am. Chem. Soc, vol.125, pp.13670-13671, 2003. ,
Environment-Independent 14-Helix Formation in Short ?-Peptides: Striking a Balance between Shape Control and Functional Diversity, Structure-activity studies of 14-helical antimicrobial beta-peptides: probing the relationship between conformational stability and antimicrobial potency, vol.3, pp.12774-12785, 2001. ,
Comparison of Design Strategies for Promotion of ?-Peptide 14-Helix Stability in Water, J. Am. Chem. Soc, vol.125, pp.2254-2259, 2003. ,
Design, machine synthesis, and NMR-solution structure of a [small beta]-heptapeptide forming a salt-bridge stabilised 3-helix in methanol and in water, J. Am. Chem. Soc, vol.0, pp.5162-5163, 2001. ,
12-Helix Formation in Aqueous Solution with Short ?-Peptides Containing Pyrrolidine-Based Residues, J. Am. Chem. Soc, vol.122, pp.4821-4822, 2000. ,
Positional screening and NMR structure determination of side-chain-to-side-chain cyclized [small beta]3-peptides, Peptide Foldamers Targeting Intracellular Protein-Protein Interactions with Activity in Living Cells, vol.10, pp.11365-11375, 2000. ,
A rapid library screen for tailoring [beta]-peptide structure and function, J. Am. Chem. Soc, vol.126, pp.14584-14585, 2004. ,
Identification of a ?3-peptide HIV fusion inhibitor with improved potency in live cells, Bioorg. Med. Chem. Lett, vol.19, pp.3736-3738, 2009. ,
Seebach, gamma-Peptides Forming More Stable Secondary Structures than alpha-Peptides: Synthesis and helical NMR-solution structure of the gamma-hexapeptide analog of H-(Val-Ala-Leu)2-OH, J. Am. Chem. Soc, vol.120, pp.983-1002, 1998. ,
Jaun, gamma2,3,4-Amino Acids, Coupling to gamma-Hexapeptides: CD Spectra, NMR Solution and X-ray Crystal Structures of gamma-Peptides, Chem. Commun, vol.8, pp.573-584, 2001. ,
Consequences of Isostructural Main-Chain Modifications for the Design of Antimicrobial Foldamers: Helical Mimics of Host-Defense Peptides Based on a Heterogeneous Amide/Urea Backbone, Angew. Chem. Int. Ed. Engl, vol.49, pp.333-336, 2010. ,
URL : https://hal.archives-ouvertes.fr/hal-00440427
Solid Phase Syntheses of Oligoureas, Stable Helical Secondary Structure in Short-Chain N,N'-Linked Oligoureas Bearing Proteinogenic Side Chains, vol.34, pp.1893-1895, 1995. ,
Folding and self-assembly of aromatic and aliphatic urea oligomers: Towards connecting structure and function, Org. Biomol. Chem, vol.8, pp.3101-3117, 2010. ,
Helix-Forming Oligoureas: Temperature-Dependent NMR, Structure Determination, and Circular Dichroism of a Nonamer with Functionalized Side Chains, Helv. Chim. Acta, vol.85, pp.3692-3711, 2002. ,
Linked Oligoureas as Foldamers: Chain Length Requirements for Helix Formation in Protic Solvent Investigated by Circular Dichroism, NMR Spectroscopy, and Molecular Dynamics, J. Am. Chem. Soc, vol.127, pp.2156-2164, 2005. ,
URL : https://hal.archives-ouvertes.fr/hal-00130006
Helix-Forming Propensity of Aliphatic Urea Oligomers Incorporating Noncanonical Residue Substitution Patterns, Condensation Approach to Aliphatic Oligourea Foldamers: Helices with N-(pyrrolidin-2-ylmethyl)ureido Junctions, vol.49, pp.4884-4892, 2010. ,
Structural characterization of short hybrid urea/carbamate (U/C) foldamers: A case of partial helix unwinding, Biopolymers (Pept Sci), vol.100, pp.687-697, 2013. ,
Mimicking Helical Antibacterial Peptides with Nonpeptidic Folding Oligomers, Chem. Biol, vol.13, pp.531-538, 2006. ,
URL : https://hal.archives-ouvertes.fr/hal-00130007
A Cell-Penetrating Foldamer with a Bioreducible Linkage for Intracellular Delivery of DNA, Angew. Chem. Int. Ed, vol.54, pp.11133-11137, 2015. ,
Stabilization of an ?-helix by short adjacent accessory foldamers, Stabilization of Short ?-Helices by Non-Peptide Helical Foldamers, vol.54, pp.123-131, 2015. ,
Sequence-specific polypeptoids: A diverse family of heteropolymers with stable secondary structure, Proc. Nat. Acad. Sci, vol.95, pp.4303-4308, 1998. ,
Extreme stability of helices formed by water-soluble poly-N-substituted glycines (polypeptoids) with ?-chiral side chains, Biopolymers, vol.63, pp.12-20, 2002. ,
Diversifying the structural architecture of synthetic oligomers: the hetero foldamer approach, Foldamers with Heterogeneous Backbones, vol.41, pp.11593-11611, 2008. ,
Stereocontrolled protein surface recognition using chiral oligoamide proteomimetic foldamers, J. Am. Chem. Soc, vol.130, pp.2434-2443, 2008. ,
/?+?)-Peptide Antagonists of BH3 Domain/Bcl-xL Recognition: Toward General Strategies for Foldamer-Based Inhibition of Protein?Protein Interactions, J. Am. Chem. Soc, vol.129, pp.335-339, 2006. ,
Surprisingly stable helical conformations in [alpha]/[beta]-peptides by incorporation of cis-[beta]-aminocyclopropane carboxylic acids, Angew. Chem. Int. Ed. Engl, vol.43, pp.505-510, 2004. ,
Residue requirements for helical folding in short [alpha]/[beta]-peptides: crystallographic characterization of the 11-helix in an optimized sequence, Angew. Chem. Int. Ed. Engl, vol.44, pp.407-429, 2005. ,
Interplay among side chain sequence, backbone composition, and residue rigidification in polypeptide folding and assembly, Proc. Nat. Acad. Sci. U.S.A, vol.105, pp.9151-9156, 2008. ,
12/10-and 11/13-mixed helices in alpha/gamma-and beta/gamma-hybrid peptides containing C-linked carbo-gamma-amino acids with alternating alpha-and beta-amino acids, Angewandte Chemie International Edition, vol.128, pp.7847-7851, 2006. ,
, Helices with Additional H-bonds: Crystallographic Conformations of ?,?-Hybrid Peptides Helices Composed of ?-Hydroxy ?-Amino acids (Statines), 2016.
Helix Formation in Preorganized ?/?-Peptide Foldamers: Hydrogen-Bond Analogy to the ?-Helix without ?-Amino Acid Residues, J. Am. Chem. Soc, vol.132, pp.7868-7869, 2010. ,
Koksch, ?-and ?-Amino Acids at ?-Helical Interfaces: Toward the Formation of Highly Stable Foldameric Coiled Coils, ACS Med. Chem. Lett, vol.9, pp.1300-1303, 2014. ,
Differential Impact of ? and ? Residue Preorganization on ?/?/?-Peptide Helix Stability in Water, J. Am. Chem. Soc, vol.133, pp.8149-8152, 2011. ,
Exploiting the Right Side of the Ramachandran Plot: Substitution of Glycines by d-Alanine Can Significantly Increase Protein Stability, Supernormal insulin: [D-PheB24]-insulin with increased affinity for insulin receptors, vol.107, pp.3852-3856, 1982. ,
Protein Design with l-and d-?-Amino Acid Structures as the Alphabet, Acc. Chem. Res, vol.41, pp.1301-1308, 2008. ,
The Gramicidin A Transmembrane Channel: A Proposed ?(L,D) Helix, Proc. Nat. Acad. Sci. U.S.A, vol.68, pp.672-676, 1971. ,
Linear stereocooligopeptides with alternating D and L residues. 3. Nature and relative stability of monomeric and dimeric species of the D,L-alternating octapeptide Boc-(L-Val-D-Val)4-OMe in cyclohexane or chloroform solution, Proc. Nat. Acad. Sci, vol.282, pp.7910-7915, 1979. ,
Engineering a ?-Helical D,L-Peptide for Folding in Polar Media, Chem. Eur. J, vol.15, pp.11867-11877, 2009. ,
Mirror image phage display -Generating stable therapeutically and diagnostically active peptides with biotechnological means, A Potent d-Protein Antagonist of VEGF-A is Nonimmunogenic, Metabolically Stable, and Longer-Circulating in Vivo, vol.271, pp.1058-1065, 1996. ,
Aromatic Oligoamide Foldamers, Aromatic Amide Foldamers: Structures, Properties, and Functions, vol.101, pp.5271-5316, 2001. ,
Novel Molecular Scaffolds: Formation of Helical Secondary Structure in a Family of Oligoanthranilamides, Angew. Chem. Int. Ed, vol.33, pp.446-448, 1994. ,
DNH deoxyribonucleohelicates: self assembly of oligonucleosidic double-helical metal complexes, Angew. Chem. Int. Ed, vol.346, pp.1838-1840, 1990. ,
Structural codons: linearity/helicity interconversion by pyridine/pyrimidine exchange in molecular strands, Proc. Natl. Acad. Sci, vol.99, pp.62-63, 2002. ,
Chiral induction in quinoline-derived oligoamide foldamers: Assignment of helical handedness and role of steric effects, Journal of the American Chemical Society, vol.127, pp.12943-12951, 2005. ,
URL : https://hal.archives-ouvertes.fr/hal-00096047
Synthesis of urea oligomers and their antibacterial activity, Biomimetic facially amphiphilic antibacterial oligomers with conformationally stiff backbones, vol.99, pp.427-435, 2002. ,
Development and Biological Assessment of Fully Water-Soluble Helical Aromatic Amide Foldamers, Angew. Chem. Int. Ed. Engl, vol.46, pp.1679-1685, 2007. ,
Solvent dependence of helix stability in aromatic oligoamide foldamers, Chem. Commun, vol.48, pp.6337-6339, 2012. ,
Solid-Phase Synthesis of Water-Soluble Helically Folded Hybrid ?-Amino Acid/Quinoline Oligoamides, J. Org. Chem, vol.81, pp.1137-1150, 2016. ,
URL : https://hal.archives-ouvertes.fr/hal-01509471
Inhibition of [alpha]-helix-mediated protein-protein interactions using designed molecules, Bioorg. Med. Chem. Lett, vol.36, pp.717-724, 2007. ,
Minimalist and universal peptidomimetics, Chem. Soc. Rev, vol.40, pp.4411-4421, 2011. ,
Toward Proteomimetics: Terphenyl Derivatives as Structural and Functional Mimics of Extended Regions of an ?-Helix, J. Am. Chem. Soc, vol.123, pp.5382-5383, 2001. ,
Development of a potent Bclx(L) antagonist based on alpha-helix mimicry, Terphenyl-Based Helical Mimetics That Disrupt the p53/HDM2 Interaction, vol.124, pp.2704-2707, 2002. ,
Terephthalamide Derivatives as Mimetics of Helical Peptides: Disruption of the Bcl-xL/Bak Interaction, Bioorg. Med. Chem. Lett, vol.14, pp.5463-5468, 2004. ,
Design and application of an alpha-helixmimetic scaffold based on an oligoamide-foldamer strategy: antagonism of the Bak BH3/Bcl-xL complex, Angew. Chem. Int. Ed. Engl, vol.42, pp.535-539, 2003. ,
Synthetic Foldamers That Mimic Extended alpha Helices ?, Angew. Chem. Int. Ed, vol.46, pp.8614-8617, 2007. ,
Oligobenzamide proteomimetic inhibitors of the p53-hDM2 proteinaprotein interaction, Tetrahedron Lett, vol.48, pp.5091-5093, 2007. ,
Synthesis of pyridazines functionalized with amino acid side chains, Synthesis of Pyridazine-Based Scaffolds as ?-Helix Mimetics, vol.49, pp.3733-3736, 2007. ,
Aromatic garlands, as new foldamers, to mimic protein secondary structure, Synthesis of new phenylpyridyl scaffolds using the Garlanding approach, vol.66, pp.2671-2680, 1910. ,
URL : https://hal.archives-ouvertes.fr/hal-00764805
A Multifaceted Secondary Structure Mimic Based On Piperidine-piperidinones, Angew. Chem. Int. Ed, vol.53, pp.4450-4458, 2014. ,
Rational Design of Topographical Helix Mimics as Potent Inhibitors of Protein-Protein Interactions, Oligooxopiperazines as Nonpeptidic ?-Helix Mimetics, vol.12, pp.7877-7888, 2010. ,
Amphiphilic [small alpha]-helix mimetics based on a benzoylurea scaffold, Novel Amphiphilic ?-Helix Mimetics Based on a Bisbenzamide Scaffold, vol.11, pp.3234-3237, 2009. ,
The Supramolecular Chemistry of ?-Sheets, J. Am. Chem. Soc, vol.135, pp.5477-5492, 2013. ,
Pleated Sheets and Turns of ?-Peptides with Proteinogenic Side Chains, Angewandte Chemie International Edition, vol.38, pp.1595-1597, 1999. ,
Antiparallel Sheet Formation in ?-Peptide Foldamers: Effects of ?-Amino Acid Substitution on Conformational Preference1, Parallel Sheet Secondary Structure in ?-Peptides, vol.119, pp.2155-2166, 1997. ,
cis-2-aminocyclopentanecarboxylic acid oligomers adopt a sheetlike structure: switch from helix to nonpolar strand, Chemical Communications, vol.114, pp.5006-5008, 1992. ,
Infinite pleated ?-sheet formed by the ?hairpin Boc-?-Phe-?-Phe-d-Pro-Gly-?-Phe-?-Phe-OMe, Peptide hybrids containing ?-and ?-amino acids: Structure of a decapeptide ?-hairpin with two facing ?-phenylalanine residues, Proc. Nat. Acad. Sci, vol.98, pp.5955-5965, 2001. ,
Hairpin Folding Behavior of Mixed ?/?-Peptides in Aqueous Solution, J. Am. Chem. Soc, vol.133, pp.4246-4249, 2011. ,
Design Strategies for the Sequence-Based Mimicry of Side-Chain Display in Protein ?-Sheets by ?/?-Peptides, J. Am. Chem. Soc, vol.134, pp.15906-15913, 2012. ,
Foldameric ?/?-Peptide Analogs of the ?-Sheet-Forming Antiangiogenic Anginex: Structure and Bioactivity, J. Am. Chem. Soc, vol.135, pp.16578-16584, 2013. ,
Introduction of Cyclically Constrained ?-Residues Stabilizes an ?-Peptide Hairpin in Aqueous Solution, Org. Lett, vol.15, pp.944-947, 2013. ,
Hydrophobic Cluster Formation Is Necessary for Dibenzofuran-Based Amino Acids to Function as .beta.-Sheet Nucleators, Hydrogen Bonded Squaramide-Based Foldable Module Induces Both ?-and ?-Turns in Hairpin Structures of ?-Peptides in Water, vol.116, pp.2980-2983, 1994. ,
Synthesis of peptide-functionalized diacylaminoepindolidiones as templates for ?-sheet formation, Tetrahedron Letters, vol.29, pp.58-66, 1988. ,
An Unnatural Amino Acid that Mimics a Tripeptide ?-Strand and Forms ?-Sheetlike Hydrogen-Bonded Dimers, J. Am. Chem. Soc, vol.122, pp.7654-7661, 2000. ,
Cyclic Modular ?-Sheets, Beta-Hairpin Peptidomimetics: Design, Structures and Biological Activities, vol.41, pp.2548-2558, 2007. ,
Amyloid ?-sheet mimics that antagonize protein aggregation and reduce amyloid toxicity, Nat Chem, vol.4, pp.927-933, 2012. ,
Let the Enzyme or Receptor be the Judge, Acc. Chem. Res, vol.44, pp.180-193, 2011. ,
Pyrrolinone-Pyrrolidine Oligomers as Universal Peptidomimetics, Journal of the American Chemical Society, vol.133, pp.12350-12353, 2011. ,
Alkyne-Linked 2,2-Disubstituted-indolin-3-one Oligomers as Extended ?-Strand Mimetics, J. Am. Chem. Soc, vol.131, pp.4566-4567, 2009. ,
A 1,3-phenyl-linked hydantoin oligomer scaffold as a [small beta]-strand mimetic, Chem. Commun, vol.48, pp.3709-3711, 2012. ,
Aryl-linked imidazolidin-2-ones as non-peptidic [small beta]-strand mimetics, Angew. Chem. Int. Ed, vol.48, pp.2649-2652, 2012. ,
Ion-mediated conformational switches, Chem. Sci, vol.6, pp.1630-1639, 2015. ,
Antiparallel side-by-side dimeric motif for sequence-specific recognition in the minor groove of DNA by the designed peptide 1-methylimidazole-2-carboxamide netropsin, Proc. Nat. Acad. Sci. U.S.A, vol.89, pp.8783-8794, 1992. ,
Recognition of the four Watson-Crick base pairs in the DNA minor groove by synthetic ligands, Nature, vol.391, pp.468-471, 1998. ,
A Structural Basis for Recognition of A·T and T·A Base Pairs in the Minor Groove of B-DNA, Science, vol.282, pp.111-115, 1998. ,
Aliphatic/Aromatic Amino Acid Pairings for Polyamide Recognition in the Minor Groove of DNA, J. Am. Chem. Soc, vol.120, pp.6219-6226, 1998. ,
Recognition of 16 Base Pairs in the Minor Groove of DNA by a Pyrrole?Imidazole Polyamide Dimer, J. Am. Chem. Soc, vol.120, pp.3534-3535, 1998. ,
Stereochemical Control of the DNA Binding Affinity, Sequence Specificity, and Orientation Preference of Chiral Hairpin Polyamides in the Minor Groove, J. Am. Chem. Soc, vol.120, pp.1382-1391, 1998. ,
Pyrrole-Imidazole Polyamides Distinguish Between Double-Helical DNA and RNA, Angew. Chem. Int. Ed, vol.52, pp.415-418, 2013. ,
Sequence-selective recognition of DNA by strand displacement with a thymine-substituted polyamide, Science, vol.254, pp.1497-1500, 1991. ,
,
PNA hybridizes to complementary oligonucleotides obeying the WatsonCrick hydrogen-bonding rules, Nature, vol.365, pp.566-568, 1993. ,
DNA unwinding upon strand-displacement binding of a thymine-substituted polyamide to double-stranded DNA, Proc. Nat. Acad. Sci, vol.90, pp.1667-1670, 1993. ,
Crystal structure of a peptide nucleic acid (PNA) duplex at 1.7 A resolution, Nat. Struct. Mol. Biol, vol.4, pp.98-101, 1997. ,
The Influence of a Chiral Amino Acid on the Helical Handedness of PNA in Solution and in Crystals, J. Biomol. Struct. Dyn, vol.21, pp.495-502, 2004. ,
Insights into peptide nucleic acid (PNA) structural features: The crystal structure of a d-lysine-based chiral PNA-DNA duplex, The Crystal Structure of Non-Modified and Bipyridine-Modified PNA Duplexes, vol.100, pp.1424-1430, 2003. ,
The first crystal structures of RNA-PNA duplexes and a PNA-PNA duplex containing mismatches-toward anti-sense therapy against TREDs, Nucleic Acids Res, vol.44, pp.1937-1943, 2016. ,
Crystal Structure of Chiral ?PNA with Complementary DNA Strand: Insights into the Stability and Specificity of Recognition and Conformational Preorganization, J. Am. Chem. Soc, vol.132, pp.10717-10727, 2010. ,
Peptide nucleic acid (PNA): its medical and biotechnical applications and promise for the future, Curr. Opin. Mol. Ther, vol.37, pp.300-303, 1998. ,
Peptide nucleic acid: a versatile tool in genetic diagnostics and molecular biology, Curr. Opin. Biotechnol, vol.12, pp.16-20, 2001. ,
Evidence from Circular Dichroism and from Melting Behavior for Helix-Inducing Complexation of a Designed ?3-Pentadecapeptide with DNA Duplexes. Preliminary Communication, Helv. Chim. Acta, vol.86, pp.3087-3103, 2003. ,
Zn2+-Complexation by a ?-Peptidic Helix and Hairpin Containing ?3hCys and ?3hHis Building Blocks: Evidence from CD Measurements. Preliminary Communication, Helv. Chim. Acta, vol.86, pp.2653-2661, 2003. ,
Structural elucidation of foldamers with no long range conformational order, Chem. Commun, vol.50, pp.10090-10093, 2014. ,
Protein-Protein Interactions Mediated by Helical Tertiary Structure Motifs, J. Am. Chem. Soc, vol.137, pp.11622-11630, 2015. ,
Targeting diverse proteinprotein interaction interfaces with ?/?-peptides derived from the Z-domain scaffold, Proc. Nat. Acad. Sci. U.S.A, vol.137, pp.4552-4557, 2015. ,
De novo design and structural characterization of proteins and metalloproteins, Annu. Rev. Biochem, vol.68, pp.779-819, 1999. ,
, ?-? linking motifs and interhelical orientations, Proteins: Structure, Function, and Bioinformatics, vol.61, pp.325-337, 2005.
De novo design and synthesis of helix-turn-helix structure from short and robust mixed helices derived from C-linked carbobeta-amino acids, Angew Chem Int Ed Engl, vol.45, pp.8207-8210, 2006. ,
Long-range interactions stabilize the fold of a non-natural oligomer, J. Am. Chem. Soc, vol.124, pp.11564-11565, 2002. ,
, A Helix?Turn?Helix Supersecondary Structure Based on Oligo, vol.10, pp.69-72, 2007.
Folding a Nonbiological Polymer into a Compact Multihelical Structure, J. Am. Chem. Soc, vol.127, pp.10999-11009, 2005. ,
Toward ?-Amino Acid Proteins: Design, Synthesis, and Characterization of a Fifteen Kilodalton ?-Peptide Tetramer, J. Am. Chem. Soc, vol.130, pp.821-823, 2008. ,
Proteomorphous objects from abiotic backbones, Angew Chem Int Ed Engl, vol.46, pp.2168-2174, 2007. ,
URL : https://hal.archives-ouvertes.fr/hal-00170390
Protein backbone engineering as a strategy to advance foldamers toward the frontier of protein-like tertiary structure, Org. Biomol. Chem, vol.12, pp.8796-8802, 2014. ,
Synthesis, folding, and structure of the ?-turn mimic modified B1 domain of streptococcal protein G, J. Am. Chem. Soc, vol.8, pp.4178-4180, 1999. ,
Artificial Chemokines: Combining Chemistry and Molecular Biology for the Elucidation of Interleukin-8 Functionality, J. Am. Chem. Soc, vol.130, pp.15311-15317, 2008. ,
Towards "bionic" proteins: replacement of continuous sequences from HIF-1[small alpha] with proteomimetics to create functional p300 binding HIF-1[small alpha] mimics, Chem. Commun, vol.52, pp.5421-5424, 2016. ,
Effects of Single ?-to-? Residue Replacements on Structure and Stability in a Small Protein: Insights from Quasiracemic Crystallization, J. Am. Chem. Soc, vol.138, pp.6498-6505, 2016. ,
Protein-like Tertiary Folding Behavior from Heterogeneous Backbones, J. Am. Chem. Soc, vol.135, pp.12528-12531, 2013. ,
Folding thermodynamics of protein-like oligomers with heterogeneous backbones, Chem. Sci, vol.5, pp.3325-3330, 2014. ,
An ?/?-Peptide Helix Bundle with a Pure ?3-Amino Acid Core and a Distinctive Quaternary Structure, J. Am. Chem. Soc, vol.131, pp.9860-9861, 2009. ,
Comparison of design strategies for [small alpha]-helix backbone modification in a protein tertiary fold, Chem. Commun, vol.52, pp.3789-3792, 2016. ,
Shaping quaternary assemblies of watersoluble non-peptide helical foldamers by sequence manipulation, Nat. Chem, vol.7, pp.871-878, 2015. ,
Improved Carbohydrate Recognition in Water with an Electrostatically Enhanced ?-Peptide Bundle, Org. Lett, vol.17, pp.4718-4721, 2015. ,
NMR-Solution Structures in Methanol of an ?-Heptapeptide, of a ?3/?2-Nonapeptide, and of an all-?3-Icosapeptide Carrying the 20 Proteinogenic Side Chains, Helv. Chim. Acta, vol.88, pp.1969-1982, 2005. ,
Residue-based control of helix shape in [beta]-peptide oligomers, Nature, vol.387, pp.381-384, 1997. ,
)-and beta(3)-peptides with proteinaceous side chains: Synthesis and solution structures of constitutional isomers, a novel helical secondary structure and the influence of solvation and hydrophobic interactions on folding, Helvetica Chimica Acta, vol.81, issue.2, pp.932-982, 1998. ,
Controlling Helix Formation in the ?-Peptide Superfamily: Heterogeneous Foldamers with Urea/Amide and Urea/Carbamate Backbones, Angew. Chem. Int. Ed, vol.52, pp.4147-4151, 2013. ,
Structural and biological mimicry of protein surface recognition by ?/?-peptide foldamers, Proc. Nat. Acad. Sci, vol.106, pp.14751-14756, 2009. ,
Iterative design of a helically folded aromatic oligoamide sequence for the selective encapsulation of fructose, Nat Chem, vol.7, pp.334-341, 2015. ,
URL : https://hal.archives-ouvertes.fr/hal-01509470
Application of microwave irradiation to the synthesis of 14-helical [beta]-peptides, Nat. Protocols, vol.7, pp.624-631, 2005. ,
Efficient method for the preparation of peptoids [oligo(N-substituted glycines)] by submonomer solid-phase synthesis, J. Am. Chem. Soc, vol.114, pp.4057-4059, 1992. ,
Microwave-Enhanced Solid-Phase Synthesis of N,N '-Linked Aliphatic Oligoureas and Related Hybrids, Org. Lett, vol.14, pp.3130-3133, 2012. ,
, Methods Enzymol, vol.580, pp.279-301, 2016.
Microwave assisted solid phase synthesis of highly functionalized N-alkylated oligobenzamide ?-helix mimetics, Bioorg. Med. Chem, vol.21, pp.4034-4040, 2013. ,
Fmoc Solid Phase Synthesis of Polyamides Containing Pyrrole and Imidazole Amino Acids, Organic Letters, vol.3, pp.1201-1203, 2001. ,
Microwave Assisted Synthesis of Py-Im Polyamides, Organic Letters, vol.14, pp.2774-2777, 2012. ,
Recent Developments of Engineered Translational Machineries for the Incorporation of Non-Canonical Amino Acids into Polypeptides, Synthesis of biopolymers using genetic code reprogramming, vol.12, pp.6513-6531, 2008. ,
Reevaluation of the d-Amino Acid Compatibility with the Elongation Event in Translation, J. Am. Chem. Soc, vol.131, pp.1830-1837, 2009. ,
, Polymerization of ?-Hydroxy Acids by Ribosomes, vol.9, pp.2773-2778, 2008.
Ribosomal Synthesis of Peptides with Multiple ?-Amino Acids, J. Am. Chem. Soc, vol.138, pp.1962-1969, 2016. ,
In Vivo Biosynthesis of a ?-Amino Acid-Containing Protein, J. Am. Chem. Soc, vol.138, pp.5194-5197, 2016. ,
The Outstanding Biological Stability of ?-and ?-Peptides toward Proteolytic Enzymes: An In Vitro Investigation with Fifteen Peptidases, ChemBioChem, vol.2, pp.445-455, 2001. ,
Peptoids: a modular approach to drug discovery, Proc. Nat. Acad. Sci, vol.89, pp.9367-9371, 1992. ,
Proteolytically Stable Foldamer Mimics of Host-Defense Peptides with Protective Activities in a Murine Model of Bacterial Infection, J. Med. Chem, vol.59, pp.8221-8232, 2016. ,
A left-handed solution to peptide inhibition of the p53-MDM2 interaction, Angew. Chem. Int. Ed. Engl, vol.49, pp.3649-3652, 2010. ,
Helical Antimicrobial Sulfono-?-AApeptides, J. Med. Chem, vol.58, pp.4802-4811, 2015. ,
, Chemistry and Biochemistry of Amino Acids, vol.7, pp.267-357, 1983.
Substrate analogues incorporating ß-amino acids: potential application for peptidase inhibition, FASEB J, 2001. ,
Cell Determinants Incorporating ?-Amino Acid Residues Are Protease Resistant and Remain Immunogenic In Vivo, J. Immunol, vol.175, pp.3810-3818, 2005. ,
The Proteolytic Stability of 'Designed' ?-Peptides Containing ?-Peptide-Bond Mimics and of Mixed ?,?-Peptides: Application to the Construction of MHC-Binding Peptides, Chem. Biodiv, vol.2, pp.591-632, 2005. ,
Antibacterial peptides for therapeutic use: obstacles and realistic outlook, Curr Opin Pharmacol, vol.6, pp.468-472, 2006. ,
Antimicrobial and host-defense peptides as new anti-infective therapeutic strategies, Nat. Biotechnol, vol.24, pp.389-395, 2002. ,
Mechanisms and consequences of bacterial resistance to antimicrobial peptides, Drug Resist. Updat, vol.26, pp.43-57, 2016. ,
De Novo Design of Antimicrobial Polymers, Foldamers, and Small Molecules: From Discovery to Practical Applications, Glycopeptide dendrimers as Pseudomonas aeruginosa biofilm inhibitors, vol.125, pp.366-415, 2003. ,
De novo design of antibacterial [beta]-peptides, J. Am. Chem. Soc, vol.121, p.565, 1999. ,
On the antimicrobial and hemolytic activities of amphiphilic beta-peptides, Chembiochem, vol.2, pp.771-773, 2001. ,
, Peptide Capable of Folding into a 12/10-Helical Secondary Structure, ChemBioChem, vol.4, pp.1345-1347, 2003.
Peptoids that mimic the structure, function, and mechanism of helical antimicrobial peptides, Proc. Nat. Acad. Sci, vol.105, pp.2794-2799, 2008. ,
Helical 1:1 ?/Sulfono-?-AA Heterogeneous Peptides with Antibacterial Activity, Biomacromolecules, vol.17, pp.1854-1859, 2016. ,
, Efficacy of Antimicrobial Peptoids against Mycobacterium tuberculosis, vol.55, pp.3058-3062, 2011.
Surfactant-facilitated crystallisation of water-soluble foldamers, Chem. Eur. J, vol.22, pp.3377-3383, 2016. ,
Unexpected relationships between structure and function in [alpha],[beta]-peptides: antimicrobial foldamers with heterogeneous backbones, J. Am. Chem. Soc, vol.126, pp.6848-6849, 2004. ,
De novo design and in vivo activity of conformationally restrained antimicrobial arylamide foldamers, Proc. Nat. Acad. Sci, vol.106, pp.6968-6973, 2009. ,
Orientation, Dynamics, and Lipid Interaction of an Antimicrobial Arylamide Investigated by 19F and 31P Solid-State NMR Spectroscopy, J. Am. Chem. Soc, vol.132, pp.9197-9205, 2010. ,
Small-molecule inhibitors of protein-protein interactions: progressing towards the dream, Small-Molecule Inhibitors of Protein-Protein Interactions: Progressing toward the Reality, vol.3, pp.1102-1114, 2004. ,
Targeting protein-protein interactions, a wide open field for drug design, C. R. Chimie, vol.19, pp.19-27, 2016. ,
Future directions for peptide therapeutics development, Drug Discov. Today, vol.18, pp.807-817, 2013. ,
Control of peptide conformation by the Thorpe-Ingold effect (C alpha-tetrasubstitution), Biopolymers, vol.60, pp.396-419, 2001. ,
An All-Hydrocarbon Cross-Linking System for Enhancing the Helicity and Metabolic Stability of Peptides, J. Am. Chem. Soc, vol.1, pp.49-75, 1995. ,
Development of ?-Helical Calpain Probes by Mimicking a Natural Protein-Protein Interaction, J. Am. Chem. Soc, vol.134, pp.17704-17713, 2012. ,
Comparative ?-Helicity of Cyclic Pentapeptides in Water, Angew. Chem. Int. Ed, vol.53, pp.6965-6969, 2014. ,
The Hydrogen Bond Mimic Approach: Solid-Phase Synthesis of a Peptide Stabilized as an α-Helix with a Hydrazone Link, Kemp, Peptidomimetics and the template approach to nucleation of ?-sheets and ?helices in peptides, vol.8, pp.3862-3875, 1990. ,
Downsizing human, bacterial, and viral proteins to short water-stable alpha helices that maintain biological potency, Hydrocarbon-Stapled Peptides: Principles, Practice, and Progress, vol.43, pp.6275-6288, 2000. ,
Beta-peptides with improved affinity for hDM2 and hDMX, Bioorg. Med. Chem, vol.17, pp.2038-2046, 2009. ,
Selective and Potent Proteomimetic Inhibitors of Intracellular Protein-Protein Interactions, Angew. Chem. Int. Ed, vol.54, pp.2960-2965, 2015. ,
First Evidence That Oligopyridines, ?-Helix Foldamers, Inhibit Mcl-1 and Sensitize Ovarian Carcinoma Cells to Bcl-xL-Targeting Strategies, J. Med. Chem, vol.58, pp.1644-1668, 2015. ,
Intermediate conformations during viral fusion glycoprotein structural transition, Annu. Rev. Biochem, vol.70, pp.143-150, 2001. ,
Peptides corresponding to a predictive alpha-helical domain of human immunodeficiency virus type 1 gp41 are potent inhibitors of virus infection, Proc. Natl. Acad. Sci. U. S. A, vol.91, pp.9770-9774, 1994. ,
Interaction between heptad repeat 1 and 2 regions in spike protein of SARS-associated coronavirus: implications for virus fusogenic mechanism and identification of fusion inhibitors, Nat. Commun, vol.363, p.5, 2014. ,
Design and characterization of ebolavirus GP prehairpin intermediate mimics as drug targets, Protein Sci, vol.24, pp.446-463, 2015. ,
Prevention of Measles Virus Infection by Intranasal Delivery of Fusion Inhibitor Peptides, Journal of Virology, vol.89, pp.1143-1155, 2015. ,
URL : https://hal.archives-ouvertes.fr/hal-01917852
Mucosal delivery of a double-stapled RSV peptide prevents nasopulmonary infection, J. Clin. Invest, vol.124, pp.2113-2124 ,
Design of helical, oligomeric HIV-1 fusion inhibitor peptides with potent activity against enfuvirtide-resistant virus, Proc. Natl. Acad. Sci. U. S. A, vol.104, pp.12772-12777, 2007. ,
Potent D-peptide inhibitors of HIV-1 entry, Proc. Nat. Acad. Sci. U.S.A, vol.104, pp.16828-16833, 2007. ,
Inhibiting HIV fusion with a beta-peptide foldamer, J. Am. Chem. Soc, vol.127, pp.13126-13127, 2005. ,
Design of a Protein Surface Antagonist Based on ?-Helix Mimicry: Inhibition of gp41 Assembly and Viral Fusion, Angew. Chem. Int. Ed, vol.41, pp.278-281, 2002. ,
Decoding and unlocking the BCL-2 dependency of cancer cells, Nat. Rev. Cancer, vol.13, pp.455-465, 2013. ,
Thirty years of BCL-2: translating cell death discoveries into novel cancer therapies, Nat. Rev. Cancer, vol.16, pp.99-109, 2016. ,
Evaluation of Diverse ?/?-Backbone Patterns for Functional ?-Helix Mimicry: Analogues of the Bim BH3 Domain, Angew. Chem. Int. Ed, vol.47, pp.315-323, 2008. ,
Potential pharmacological chaperones targeting cancer-associated MCL-1 and Parkinson diseaseassociated ?-synuclein, Proc. Nat. Acad. Sci, vol.111, pp.11007-11012, 2014. ,
Inhibiting the p53-MDM2 interaction: an important target for cancer therapy, Targeting protein-protein interactions: Lessons from p53/MDM2, vol.8, pp.25-37, 2003. ,
, Structure of the MDM2 oncoprotein bound to the p53 tumor suppressor transactivation domain, vol.274, pp.948-953, 1996.
A small synthetic peptide, which inhibits the p53-hdm2 interaction, stimulates the p53 pathway in tumour cell lines, J. Mol. Biol, vol.299, pp.245-253, 2000. ,
Aib-based peptide backbone as scaffolds for helical peptide mimics, J. Pept. Res, vol.60, pp.88-94, 2002. ,
Reactivation of the p53 tumor suppressor pathway by a stapled p53 peptide, J. Am. Chem. Soc, vol.129, pp.2456-2457, 2007. ,
, A Stapled p53 Helix Overcomes HDMX-Mediated Suppression of p53, vol.18, pp.411-422, 2010.
, High Specificity in Protein Recognition by Hydrogen-Bond-Surrogate ?-Helices: Selective Inhibition of the p53/MDM2 Complex, vol.11, pp.2104-2107, 2010.
, Miniature Protein Inhibitors of the p53-hDM2 Interaction, vol.7, pp.29-31, 2006.
Solution structure of a [beta]-peptide ligand for hDM2, J. Am. Chem. Soc, vol.127, pp.4118-4119, 2005. ,
In Silico Improvement of beta3-peptide inhibitors of p53 x hDM2 and p53 x hDMX, J Am Chem Soc, vol.131, pp.6356-6357, 2009. ,
Cell-Permeable ?-Peptide Inhibitors of p53/hDM2 Complexation, ChemBioChem, vol.10, pp.990-993, 2009. ,
Intrinsically Cell-Permeable Miniature Proteins Based on a Minimal Cationic PPII Motif, J. Am. Chem. Soc, vol.129, pp.14578-14579, 2007. ,
Nucleation Effects in Peptide Foldamers, J. Am. Chem. Soc, vol.134, pp.11495-11502, 2012. ,
Dpeptide inhibitors of the p53-MDM2 interaction for targeted molecular therapy of malignant neoplasms, Proc. Natl. Acad. Sci. U. S. A, vol.107, pp.14321-14326, 2010. ,
Design, Synthesis, and Evaluation of an ?-Helix Mimetic Library Targeting Protein?Protein Interactions, J. Am. Chem. Soc, vol.131, pp.5564-5572, 2009. ,
, Org. Biomol. Chem, vol.10, pp.6469-6472, 2012.
, Org. Biomol. Chem, vol.8, pp.2344-2351, 2010.
, Methods Enzymol, vol.487, pp.545-574, 2011.
Adding Diverse Noncanonical Backbones to Rosetta: Enabling Peptidomimetic Design, PLoS ONE, issue.8, p.67051, 2013. ,
, Small-Molecule Proteomimetic Inhibitors of the HIF-1?-p300 Protein-Protein Interaction, vol.15, pp.1083-1087, 2014.
Affibody molecules: Engineered proteins for therapeutic, diagnostic and biotechnological applications, FEBS Letters, vol.584, pp.2670-2680, 2010. ,
Solution structure of a phage-derived peptide antagonist in complex with vascular endothelial growth factor1, J. Mol. Biol, vol.316, pp.839-845, 2002. ,
Extending Foldamer Design beyond ?-Helix Mimicry: ?/?-Peptide Inhibitors of Vascular Endothelial Growth Factor Signaling, J. Am. Chem. Soc, vol.134, pp.7652-7655, 2012. ,
Generation of tumour-necrosis-factor-?specific affibody1 molecules capable of blocking receptor binding in vitro, Biotechnol. Appl. Biochem, vol.54, pp.93-103, 2009. ,
, A synthetic IgG-binding domain based on staphylococcal protein A, Protein Eng, vol.1, pp.107-113, 1987.
High-resolution solution NMR structure of the Z domain of staphylococcal protein A1, J. Mol. Biol, vol.272, pp.573-590, 1997. ,
Chemical synthesis and X-ray structure of a heterochiral {D-protein antagonist plus vascular endothelial growth factor} protein complex by racemic crystallography, Proc. Nat. Acad. Sci, vol.109, pp.14779-14784 ,
Passing the baton in class B GPCRs: peptide hormone activation via helix induction?, Trends Biochem. Sci, vol.34, pp.303-310, 2009. ,
Chemical modification of Class II G protein-coupled receptor ligands: Frontiers in the development of peptide analogs as neuroendocrine pharmacological therapies, Pharm. Ther, vol.125, pp.39-54, 2010. ,
Insights into the structure of class B GPCRs, Trends in Pharmacological Sciences, vol.35, pp.12-22, 2014. ,
Parathyroid Hormone (PTH)-(1â?"14) and -(1â?"11) Analogs Conformationally Constrained by α-Aminoisobutyric Acid Mediate Full Agonist Responses via the Juxtamembrane Region of the PTH-1 Receptor, Proc. Natl. Acad. Sci. U. S. A, vol.92, pp.6412-6420, 1995. ,
Backbone modification of a polypeptide drug alters duration of action in vivo, Nat. Biotech, vol.32, pp.653-655, 2014. ,
Backbone Modification of a Parathyroid Hormone Receptor-1 Antagonist/Inverse Agonist, ACS Chemical Biology, 2016. ,
A Potent ?/?-Peptide Analogue of GLP-1 with Prolonged Action in Vivo, J. Am. Chem. Soc, vol.136, pp.12848-12851, 2014. ,
Characteristics of Amyloid-Related Oligomers Revealed by Crystal Structures of Macrocyclic ?-Sheet Mimics, Proc. Nat. Acad. Sci. U.S.A, vol.133, pp.6736-6744, 2011. ,
Specific aromatic foldamers potently inhibit spontaneous and seeded A?42 and A?43 fibril assembly, Biochem. J, vol.464, pp.85-98, 2014. ,
A Peptidomimetic Approach to Targeting Pre-amyloidogenic States in Type II Diabetes, Synthetic ?-Helix Mimetics as Agonists and Antagonists of Islet Amyloid Polypeptide Aggregation, vol.16, pp.736-739, 2009. ,
Folded Small Molecule Manipulation of Islet Amyloid Polypeptide, Chem. Biol, vol.21, pp.775-781, 2014. ,
Foldamer-mediated manipulation of a pre-amyloid toxin, Nat. Commun, 2016. ,
Protein transduction: unrestricted delivery into all cells?, Trends Pharmacol. Sci, vol.21, pp.290-295, 2000. ,
Cell-Penetrating Peptides: Design, Synthesis, and Applications, Fifteen Years of Cell-Penetrating, Guanidinium-Rich Molecular Transporters: Basic Science, Research Tools, and Clinical Applications, vol.8, pp.2944-2954, 1972. ,
The design, synthesis, and evaluation of molecules that enable or enhance cellular uptake: Peptoid molecular transporters, Proc. Nat. Acad. Sci, vol.97, pp.13003-13008, 2000. ,
Enantiomeric and Diastereoisomeric (Mixed) L/ D-Octaarginine Derivatives -A Simple Way of Modulating the Properties of Cell-Penetrating Peptides, Chem. Biodiv, vol.10, pp.1165-1184, 2013. ,
Cellular uptake and membrane-destabilising properties of ?-peptide/?-peptoid chimeras: lessons for the design of new cell-penetrating peptides, Biochim. Biophys. Acta -Biomembranes, vol.1778, pp.2487-2495, 2008. ,
Novel Cell-Penetrating Peptides Based on ?-Aminoxy Acids, ChemBioChem, vol.13, pp.73-79, 2012. ,
Oligocarbamate molecular transporters: Design, synthesis, and biological evaluation of a new class of transporters for drug delivery, J. Am. Chem. Soc, vol.124, pp.13382-13383, 2002. ,
Garc??a-Echeverr??a, S. Ruetz, ?-Homolysine Oligomers: A New Class of Trojan Carriers, Chemical and Biological Investigations of ?-Oligoarginines, vol.3, pp.65-97, 2002. ,
HeLa Cell Entry by Guanidinium-Rich ?-Peptides: Importance of Specific Cation-Cell Surface Interactions, J. Am. Chem. Soc, vol.127, pp.917-926, 2005. ,
A preorganized ?-amino acid bearing a guanidinium side chain and its use in cell-penetrating peptides, Org. Biomol. Chem, vol.13, pp.5617-5620, 2015. ,
Histidine-rich amphipathic peptide antibiotics promote efficient delivery of DNA into mammalian cells, Proc. Natl. Acad. Sci, vol.100, pp.1564-1568, 2003. ,
Inhibition of vascular endothelial growth factor with a sequence-specific hypoxia response element antagonist, Proc. Nat. Acad. Sci. U.S.A, vol.101, pp.16768-16773, 2004. ,
Modulation of NF-?B-dependent gene transcription using programmable DNA minor groove binders, Proc. Nat. Acad. Sci, vol.109, pp.1023-1028 ,
Deciphering Aromatic Oligoamide Foldamer-DNA Interactions, Angew. Chem. Int. Ed, vol.51, pp.473-477, 2012. ,
The outstanding metabolic stability of a 14C-labeled ?-nonapeptide in rats -in vitro and in vivo pharmacokinetic studies, Biopharm. Drug Dispos, vol.23, pp.251-262, 2002. ,
, Vivo Biodistribution and Small Animal PET of 64Cu-Labeled Antimicrobial Peptoids, vol.23, pp.1069-1079, 2012.
ADME Investigations of Unnatural Peptides: Distribution of a 14C-Labeled ? 3-Octaarginine in Rats, Chem. Biodiv, vol.4, pp.1413-1437, 2007. ,
Pharmacokinetic Modeling and Prediction of Plasma Pyrrole-Imidazole Polyamide Concentration in Rats Using Simultaneous Urinary and Biliary Excretion Data, Biol. Pharm. Bull, vol.32, pp.8471-8476, 2009. ,
Transcriptional inhibition of progressive renal disease by gene silencing pyrrole-imidazole polyamide targeting of the transforming growth factor-?1 promoter, Proc. Nat. Acad. Sci, vol.79, pp.1863-1868, 2013. ,
, Vivo, In Vitro, and In Silico Characterization of Peptoids as Antimicrobial Agents, vol.11, p.135961, 2016.
Animal models of human anthrax: the Quest for the Holy Grail, Mol Aspects Med, vol.30, pp.467-480, 2009. ,
Selective VIP Receptor Agonists Facilitate Immune Transformation for Dopaminergic Neuroprotection in MPTP-Intoxicated Mice, J. Neuroscience, vol.35, pp.16463-16478, 2015. ,
Terephthalamide derivatives as mimetics of helical peptides: disruption of the Bclx(L)/Bak interaction2005, vol.127, pp.5463-5468 ,
Targeted delivery of a novel palmitylated D-peptide for antiglioblastoma molecular therapy, Journal of Drug Targeting, vol.20, pp.264-271, 2012. ,
Melanoma peptide MART-1(27-35) analogues with enhanced binding capacity to the human class I histocompatibility molecule HLA-A2 by introduction of a beta-amino acid residue: Implications for recognition by tumor-infiltrating lymphocytes, A Novel Retro-Inverso Gonadotropin-Releasing Hormone (GnRH) Immunogen Elicits Antibodies That Neutralize the Activity of Native GnRH, vol.39, pp.3262-3269, 1999. ,
Efficient binding of reduced peptide bond pseudopeptides to major histocompatibility complex class I molecule, J Biol Chem, vol.270, pp.26057-26059, 1995. ,
Partially modified retro-inverso pseudopeptides as non-natural ligands for the human class I histocompatibility molecule HLA-A2, J Med Chem, vol.39, pp.200-208, 1996. ,
Heteroclitic properties of mixed ?-and aza-?3-peptides mimicking a supradominant CD4 T cell epitope presented by nucleosome, Mol. Immunol, vol.44, pp.3024-3036, 2007. ,
URL : https://hal.archives-ouvertes.fr/hal-00326619
Consequences of Periodic ?-to-?3 Residue Replacement for Immunological Recognition of Peptide Epitopes, ACS Chem. Biol, vol.10, pp.844-854, 2015. ,
, HIF-1?, pp.816-826